From: ImmunoPET imaging of amyloid-beta in a rat model of Alzheimer’s disease with a bispecific, brain-penetrating fusion protein
Radioligand
Reaction yield (%)
Molar activity (MBq/nmol)
[124I]I-OX265F(ab′)2Bapi
57.0 ± 6.9
60.0 ± 24.2
[125I]I-OX265F(ab′)2Bapi
21.6 ± 11.2
26.5 ± 26.6
[124I]I-OX2676F(ab′)2Bapi
58.5 ± 3.1
209.1 ± 5.9